Final programme - Posters sessions
Programme and abstracts for poster session - download HERE
| S02P | Structure and dynamics of cholinesterases and OP hydrolases |
| S02P-1 | 3D structure of natural tetrameric form of human butyrylcholinesterase obtained by Cryo-electron microscopy Konstanin M. Boyko |
| S02P-2 | Butyrylcholinesterase-proteins interactions in human blood serum Jacek Jasiecki |
| S02P-3 | Dimerization interface of cholinesterases: analysis of crystal structures, free energy molecular dynamics calculations,and in silico alanine screening Novichkova D. A. |
| S03P |
Interaction of cholinesterases with substrates, inhibitors and reactivators
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| S03P-1 | 4-aminoquinolines as reversible inhibitors of human cholinesterase activity Anita Bosak |
| S03P-2 | Synthesis of Nerve Agents’ surrogates from Dialkyl Alkylphosphonates for Antidote Screening and Toxicological Studies Samir F. de A. Cavalcante |
| S03P-3 | Biological evaluation of cysteine targeted insecticides Hrabinova M., Schmidt M. |
| S03P-4 | An alternative substrate for human erythrocyte Acetylcholinesterase activity detection Sheemona Chowdhary |
| S03P-5 | Acetylcholinesterase reactivators based on oxime-functionalized biodegradable ionic liquids Yevgen Karpichev |
| S03P-6 | In silico screening of novel BChE-reactivators Tomas Kucera |
| S03P-7 | Phenyltetrahydroisoquinoline-based triazole compounds are high-affinity potential reactivators of nerve agent-inhibited human acetylcholinesterase Nikolina Maček Hrvat |
| S03P-8 | In silico and In vitro evaluation of two novel oximes K456 and K733 against paraoxon inhibited human acetylcholinesterase and butyrylcholinesterase Syed M Nurulain |
| S03P-9 | Facile synthesis of cysteine-acetylcholinesterase targeted insecticides Miroslav Psotka |
| S03P-10 | Inhibition of human acetylcholinesterase and butyrylcholinesterase by methylene violet 3RAX Seda Onder |
| S03P-11 | Molecular modeling studies on the interactions of aflatoxin B1 and its metabolites with pheripheral and catalytic anionic sites of human acetylcholinesterase Joyce S. F. D. de Almeida |
| S03P-12 | Chlorinated pyridinium oximes are potent reactivators of acetylcholinesterase inhibited by nerve agents Tamara Zorbaz |
| S03P-13 | Expi 293 cells expressing an endogenous wild-type butyrylcholinesterase, and a variety of esterases that self-reactivates after phosphylation by all types of organophosphorus agents Irina Zueva |
| S03P-14 | Bistable dynamic behavior of endogenous butyrylcholinesterase expressed in Expi293 cells Irina Zueva |
| S04P | Reactivators of AChE, OP inhibitors - mechanism of toxicity, detection and analytical methods, diagnosis of exposure, detoxification and therapy; counter-terrorism strategies |
| S04P-1 | Reactivating efficacy of oximes K203 and K027 against a direct acetylcholinesterase inhibitor in rat diaphragm: dose-response modeling Evica Antonijevic |
| S04P-2 | Inhibition of cholinesterases following percutaneous intoxication with V agents in rats Jiri Bajgar |
| S04P-3 | Near attack conformation approach for molecular modeling studies upon the prophylactic agent 7-methoxytacrine-4-pyridinealdoxime hybrid compared with other reactivators of VX-inhibited HssAChE Tanos Celmar Costa França |
| S04P-4 | Design, synthesis and in vitro evaluation of a promising new class of bifunctional uncharged hybrid reactivators for nerve agent-inhibited human acetylcholinesterase José Dias |
| S04P-5 | The early tissue alteration induced by different oximes in rats Vesna Jaćević |
| S04P-6 | Cytotoxicity study of oxime@CB7 complexes for central nervous system penetration of quaternary acetylcholinesterase reactivators Petr Jost |
| S04P-7 | Brain Exposure of bis-Pyridinium Oxime KR-26256 Young-Sik Jung |
| S04P-8 | Analysis of bis-pyridinium mono-aldoximes in serum and organs using a high-throughput high performance liquid chromatography approach Gellert Karvaly |
| S04P-9 | A comparison of the reactivating and therapeutic efficacy of a novel bispyridinium oxime K870 with commonly used pralidoxime and the oxime HI-6 in sarin-poisoned rats and mice Jiri Kassa |
| S04P-10 | The monoquarternary reactivators for the treatment of organophoshorous intoxication Korabecny J. |
| S04P-11 | Decontamination of warfare agent Jan Marek |
| S04P-12 | In vitro characterization of the standard acetylcholinesterase reactivators Muckova L., Hepnarova V. |
| S04P-13 | Uncharged Reactivators of Cholinesterases Inhibited by Organophosphorus Nerve Agents N. Probst |
| S04P-14 | In vitro determination of oxidative stress induced by oxime reactivators using chromatographic methods Váňova N. |
| S04P-15 | In vitro evaluation of quinuclidinium oximes as reactivators of human cholinesterases inhibited by organophosphorus compounds Antonio Zandona |
| S05P | Enzymes and proteins other than ChEs interacting with OP |
| S05P-1 | Determination of BChE Activity by Mass Spectrometric Analysis of Its Adduct with Russian Vx Murashko E.A. |
| S05P-2 | An in-vitro induction of Paraoxonase 3 activity in Hepatocytes by Resveratrol Kumari Priyanka |
| S06P | Stoichiometric bioscavanger, biotechnology and therapeutical aspects |
| S06P-1 | Smart & Innovative Tools for Cholinesterases Related Applications Emilie David |
| S06P-2 | In Vitro Evaluation of Standard Acetylcholinesterase Reactivators as Reactivators of Human Plasma Butyrylcholinesterase Lucie Junova |
| S06P-3 | Novel bisquaternary heteroaromatic compounds as potential reactivators of human butyrylcholinesterase David Malinak, Eugenie Nepovimova |
| S09P | Biological functions, development and non-cholinergic function of cholinesterases |
| S09P-1 | Butyrylcholinesterase and its variants (rs3495 & rs1803274) association with Major Depressive Disorder Sliha Awan |
| S09P-2 | Alkaloids derived from traditional Chinese medicine are inhibitors for inflammation and acetylcholinesterase Xiang P. Kong |
| S09P-3 | Acetylcholinesterase regulates inflammatory responses in cultured macrophages: a player in cholinergic anti-inflammatory pathway Etta Y. L. Liu |
| S09P-4 | Genistein, a phytoestrogen in soybean, induces the expression of acetylcholinesterase via G protein-coupled receptor 30 in PC12 cells Etta Y. L. Liu |
| S09P-5 | Status of Cholinesterases in Heroin, Hashish (Cannabis) and Polydrug Addicts Syed M Nurulain |
| S09P-6 | Indirect effects of dioxin on neuronal AChE expression via astrocytes Rui Sha |
| S09P-7 | Non-neuronal cholinergic system in rat aorta Szmicseková K. |
| S09P-8 | Microphthalmia-associated transcription factor regulates acetylcholinesterase expression during melanogenesis of B16F10 cells: a cholinergic regulator in pigmentation Qiyun Wu |
| S10P | Alzheimer's disease and diseases related to cholinesterases |
| S10P-1 | Dual binding site inhibitors of acetylcholinesterase as therapeutic treatments for Alzheimer’s disease: any need for an update? K. Petrov |
| S10P-2 | Detection of Alzheimer’s drug candidate by Surface-Enhanced Raman Spectroscopy Jan Proska |
| S11P | Multi-target-directed ligands in Alzheimer's disease primarily targeting cholinesterases |
| S11P-1 | Butyrylcholinesterase inhibitors grafted with antioxidant and neuroprotective activities: novel multifunctional ligands for Alzheimer’s disease Damijan Knez |
| S11P-2 | 7-MEOTA-donepezil hybrids: Potential cholinesterase inhibitors for the treatment of Alzheimer’s disease Katarina Spilovska |